N'ime ọgwụ ndị na-anụ ma na-akpata ọgba aghara, otu n'ime ebe mbụ ka meldonia, ihe na-eme ọ bụghị nanị ndị dọkịta na ndị ọrịa, kamakwa ndị na-eme egwuregwu, ndị agha na ndị nkịtị bụ ndị na-enweghị nsogbu ahụike pụrụ iche. Ihe maka meldonium, ihe ga-eme mgbe ọ natara ya, anyị ga-atụle n'ihu.
Meldonius - gini bu ogwu a?
Meldonium na-emejupụta meldonium (Mildronate - aha ahia) na narị afọ asaa nke narị afọ gara aga site n'aka onye ọkà mmụta sayensị Latvian Kalvinshem na e jiri ya mee ihe n'ubi iji mee ka ụmụ anụmanụ na anụ ọkụkọ na osisi too. Ihe abuo bu ihe anaghi emeputa nke gamma-butyrobetaine, nke bu carnitine, ihe a na-eme n'ime ahu maka ihe di mkpa. Otu n'ime ọrụ nke carnitine bụ ihe metụtara usoro na-emetụta ụbụrụ na-agụnye ịkwafe abụba abụba n'ime sel ahụ, ebe a na-eme ka abụba ghọọ ike.
Kemgbe afọ 1984, meldoonia, a na-arụ ọrụ ahụ nke a na-amụ ruo taa, malitere itinye ya na ọgwụ. N'afọ 2012, e tinyere ya na ndepụta ọgwụ ndị dị mkpa na Russia, na 2015, World Anti-Doping Agency amachibidoro ọgwụ a iji mee ihe na egwuregwu ndị ọkachamara (ndị nchọpụta si mba ọzọ ekpebiwo na meldonium na-agbada). Taa, ọgwụ dị na pharmacies na ụdị atọ: capsules, syrup na ngwọta maka injections.
Meldonium - ụkpụrụ nke ihe
Anyị ga-achọpụta mmetụta mmetụta nke muldonium nwere n'ahụ ahụ. Ebe ọ bụ na onyinye a, ịbụ ihe yiri nke gamma-butyrobetaine, nwere ike ime ka ọnụ ọgụgụ nke carnitine pụta, nke a na-agụnye nkwụsị nke usoro ịfefe abụba na sel sel. Mmetụta a dị ezigbo mkpa n'oge oge ikuku ikuku oxygen na-enweta, ebe ọ bụ na ọ na-ejikarị abụba abụba na eriri oxygen na-emekọ ihe, enweghi ọgwụgwọ zuru oke nke abụba abụba na-emepụta ihe ndị na-emerụ ahụ maka obi.
Tinyere ngwa ngwa nke metabolism nke acid fatty acid n'okpuru ndu nke meldonia enwekwuwanye na ọnụ ọgụgụ nke mmanụ aṅụ na-emepụta, nke na-achọ ihe oriri nke oxygen. N'ihi nke a, ịrụ ọrụ nke ọma nke ATP (isi ike), na-eme ka nghazi dị n'etiti mkpa nke sel na oxygen na nnyefe ya na ọbara, kpochapụ nchịkọta nke ogige ndị na-egbu egbu n'ime sel.
Na mgbakwunye, tinyere usoro ndị a, a na-ahụwanye mmụba nke gamma-butyrobetaine, nke nwere ọdịdị ọdịdị. Nke a na-eme ka ahụ dị jụụ nke arịa ọbara ahụ, na-agbanyekwu ọkụ nke arịa ọbara, na-eme ka ọbara gbanwee, nke a na-eduzi n'akụkụ ebe ndị ahụ.
Ka anyi deputa isi ihe kachaa emetuta ya na iketa Meldonia:
- njirịta ozi;
- ọgwụ antihypoxic;
- nnyeòhèrè ọrụ
- nkwụsịtụ;
- mmelite nke mgbasa ọbara;
- mmetụta ụbụrụ;
- enwekwu ntachi obi, ike ịrụ ọrụ;
- mweghachi nke nchekwa ike n'oge na-adịghị anya;
- belata oke mgbaàmà nke mgbagha uche na nke anụ ahụ;
- normalization nke nsogbu cellular;
- iwepụ mmanya na-ewepụ mmanya.
Kedu ihe bụ meldonium?
N'iburu mmetụta dị n'ahụ meldonium ahụ, ọ bụ ihe amamihe dị na ya iji ya maka ọnọdụ dị iche iche metụtara ikuku oxygen na ụba nchekasị. Ọtụtụ mgbe, maka ọgwụgwọ ahụ, ọgwụ a abụghị ọgwụ bụ isi ma anaghị eji ya iche, ma edere ya dịka akụkụ nke ọgwụ zuru ezu. Meldonia agba akaebe na nkà mmụta ọgwụ nwere ihe ndị a:
- ọrịa obi na-adịghị ala ala;
- ọrịa na-edozi ahụ;
- nkwonkwo myocardial;
- angina pectoris;
- dystrophy myocardial;
- mmebi nke ịrụ ọrụ nke usoro obi nke usoro ihe arụ n'oge uto;
- neurocirculatory dystonia na-eto eto;
- ụbụrụ nke ụbụrụ;
- nkwupụta ụbụrụ;
- ọrịa anya na-ekesa na ọbara na-adịghị mma n'ahụ anya;
- ọbara ọbara n'ime anya nke anya;
- thrombosis nke akwa vein ma ọ bụ alaka nke anya azụ;
- retinopathy nke ọrịa mamịrị ma ọ bụ hypertensive sitere;
- abstinence mmanya;
- ihe omimi nke usoro iku ume, tinyere ude oxygen (bronchitis na-adịghị ala ala, ụkwara ume ọkụ);
- belata n'iche echiche ma ọ bụ nke anụ ahụ dị iche iche;
- Oge mmechi mgbe ọgbụgba dịgasị iche iche.
Meldonium - ngwa
Jiri meldonium na mbadamba, sirop ma ọ bụ na-egbu ogwu (na intravenously, intramuscularly or parabulbar - mmebata site na anụ nke ala nkuchianaya). A na-ekpebi ihe dị iche iche, ogologo oge na oge nke ikuku, n'otu n'otu, dabere na nyocha na oke nke ọnọdụ onye ọrịa ahụ. Okwesiri ighota na apughi imeri ọgwụ ahu n'emeghi nzube ahuike, n'ihi na ndigichi nke aka na aru nke obi, mmebi nke metabolism nke sitere na okike nwere ike inwe nsogbu njo.
Meldonium maka ndị na-eme egwuregwu
N'ịmara mmetụta muldonia nwere ike inwe n'ahụ, ọ ga-edozi ihe mere ndị egwuregwu jiri ya. A na-eji ngwá ọrụ ahụ eme ihe nile dị iche iche nke egwuregwu: egwuregwu, ịgba chaa chaa, bọllon, mgba, ozubu, igwu mmiri na ndị ọzọ. Eji Mildronate n'egwuregwu iji nweta ihe ndị na-esonụ:
- mgbochi nchịkọta n'ime mkpụrụ ndụ nke ngwaahịa na-emerụ emerụ nke abụba abụba a na-ekwughị;
- ndozi nke ike na-arụ ọrụ n'ime mkpụrụ obi obi na mmelite nke ha na-agafe;
- ịkwalite ịkwalite nsụgharị myocardial;
- meziwanye ahụ ike;
- na-amụbawanye ike na ọzụzụ nke ọzụzụ;
- ike ọgwụgwụ;
- mmelite nke mgbake nke ahu mgbe omumu.
Ọnụ ọgụgụ kwa ụbọchị nke ọgwụ maka ndị na-eme egwuregwu bụ 15-20 mg kwa kilogram nke arọ dị n'ụdị capsule. A na-atụ aro ka ị jiri ọgwụ ahụ ruo 30-40 nkeji tupu mmalite nke mgbatị ahụ. Usoro nke nnyefe sitere na otu ruo ọnwa ndị ahụ, mgbe nke ahụ gasịrị, ị ga-eme mkpọtụ maka ọbụlagodi ọnwa 1. A nabatara meldonium asọmpi n'ime izu abụọ, na n'oge asọmpi - ọ bụghị karịa ụbọchị 14. N'oge ahụ, a machibidoro ọgwụ ahụ na nnukwu egwuregwu, na ndị na-eso ya, bụ ndị a hụrụ ọbara ha, a na-emezigharị ya.
Mkpụrụ obi na ọrịa shuga
N'oge na-adịbeghị anya, e jiriwo ụdị ọnụọgụ abụọ maka ụdị ọrịa shuga na ụdị 1, nke dabeere na nchọpụta nke gosiri na o nwere ike iji ihe dị arọ belata glucose n'ime ọbara. N'otu oge ahụ, ịta insulin adịghị arị elu. Ọtụtụ mgbe, ọrịa a, a na-eji ọgwụ ahụ eme ihe na iji metformin (onye na-ebute shuga na-esite na nnukwu ụlọ). Ọgwụgwọ dị otú ahụ, na mgbakwunye na ịbelata shuga shuga, na-enye mmetụta ndị a:
- igbochi nkwụsịtụ endothelial na ọnwụ nke inwe mmetụta uche na mgbu;
- nkwado nke obi obi, mweghachi nke usoro metabolic n'ime ya;
- igbochi mmepe nke ịrịa ọrịa shuga, neuropathy na oke ibu;
- mgbochi nke ọnya-azu.
Meldonias na arrhythmia nke obi
Ọ bụrụ na ọkpụkpụ obi na-arụ ọrụ na-ezighị ezi, a na-agbaji ụda obi dị mma - arrhythmia. N'okwu a, ndị ọkachamara nwere ike ịkwado meldonium, ngwa na nkà mmụta ọgwụ nke na-egosi ezigbo nsonaazụ. Mgbe ị na-eji ọgwụ ọjọọ eme ihe na mgbagwoju anya, ọ ga-ekwe omume iji nweta nchedo siri ike nke ụda obi. N'ihi ịṅụ ọgwụ na ndị ọrịa, ihe ize ndụ nke ịmepụta angina pectoris , obere mgbatị mịnchide na -ebelata.
Meldonium si nrụgide
Meldonium, nke mmetụta ya na ahụ gosipụtara onwe ya karia na usoro nke usoro obi, ga-aba uru nye ndị nwere ọbara mgbali elu. Nnyocha na-egosi na ọgwụ ahụ, tinyere ọrịa ọgwụgwọ kachasị (n'etiti nke bụ mmetụta dị mkpa nke vasodilating maka ibelata nrụgide), na-enyere aka belata ọkwa ọkwa cholesterol n'ọbara - ihe kpatara ọbara mgbali elu. N'okwu a, a pụrụ ịgwa ndị ọrịa ka ha jiri meldonium intramuscularly mee ihe.
Meldonium na aṅụrụma
Mmiri meldonia dị mma site na nkwụsi ike , ngosipụta nke mgbaàmà nkwụsị na ndị ọrịa na-aṅụbiga mmanya ókè. Ọgwụ ọ bụghị nanị na ọ dị mma, kama ọ na-egbochi nkwụsị nke nnukwu nsogbu ndị metụtara mmanya na-aba n'obi na ụbụrụ. Onu ogugu di otu a bu ihe mgita 500, nke na-ewe 3-4 ugboro kwa ubochi maka 7-10. A na-enwe usoro ọmụmụ ọgwụgwọ n'oge etiti nke ọbụlagodi ọnwa 1-2.
Meldoniy si ike
N'ọnọdụ ụfọdụ, a na-ahọrọ meldoniy na-agwọ ọrịa maka ike ọgwụgwụ na-adịghị agwụ agwụ na-enwe mmetụta nke nchekasị uche na uche, na mgbe ahụ gwụchara n'ihi ọrịa na-adịte aka. Ọgwụ ọjọọ, nke nwere mmetụta dị mma tonic, na-enyere ahụ aka ịnagide nrụgide na-enweghị mmebi nke usoro obi, kama na-agbake, wepụ adịghị ike na ụra.
Meldonium - mmetụta ndị dị na ya
Ka anyị kọwaa ihe mmetụta ọjọọ meldoniy nwere ike ịkpasu iwe:
- overexcitation, ọgba aghara;
- isi ọwụwa;
- oke igwe;
- ụda na ntị;
- egwu;
- ike ọgwụgwụ nke uche;
- a na-atụ egwu;
- gbanwee ọbara mgbali;
- tachycardia;
- obi erughị ala;
- pallor ma ọ bụ hypremia;
- dyspepsia;
- ụkwara;
- ezigbo uto na ọnụ;
- ọnụ mmiri;
- abdominal mgbu;
- afọ ọsịsa;
- nkwonkwo akwara;
- ọzịza;
- mmeghachi omume na-ekesa (ọkụ ọkụ, itching, Quincke's edema) na ndị ọzọ.
Ndi mulberry eji ya?
A chọpụtara na meldonium na Mildronate, nke eji ogologo oge mee ihe, na-eri ahụ ụfọdụ. Ihe kachasị mma bụ mmetụta ọjọọ nke ndị na-eme egwuregwu, bụ ndị, mgbe ha kwụsịrị iji ọgwụ ọjọọ eme ihe, malite ịmalite nsogbu nsogbu uche - mmetụta nke enweghị njikere maka ọzụzụ ma ọ bụ asọmpi, ike ọgwụgwụ, adịghị ike.
Meldonium - contraindications maka ojiji
Nkọwa ọgwụgwọ meldonium contraindications ka ọkwa ahụ nwere ihe ndị a:
- onye ọ bụla na-enwe mmetụta maka akụkụ nke ọgwụ ahụ;
- nrụgide intracranial ka njọ;
- mgbatị ma ọ bụ ọgwụgwọ na-ezughị ezu, siri ike;
- afọ ime, oge ị na-aṅụ ara.
Meldonium - ihe analogues nke nkwadebe
Ọ bụrụ na ọ gaghị ekwe omume iji ọgwụ ọjọọ eme ihe nwere meldonium, a pụrụ iji analogues na-egosipụta ụdị ọgwụ ahụ yiri nke ahụ na nkwekọrịta. Ụdị ọgwụ ndị a gụnyere:
- Dibikor;
- Vero-Riboxin;
- Nyocha;
- Coenzyme Q10;
- Lipamid;
- Riboxin .